Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T72274 |
IACS-9571 hydrochloride
ASIS-P040 hydrochloride |
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IACS-9571 (ASIS-P040) hydrochloride 是溴结构域蛋白 TRIM24和 BRPF1的抑制剂,对 TRIM24 的 IC50和 Kd 值分别为 8 nM 和 31 nM,对 BRPF1的 Kd 值为 14 nM。 | |||
T11597L |
IACS-9571 Hydrochloride (1800477-30-8 free base)
IACS-9571 Hydrochloride,ASIS-P040 Hydrochloride |
Epigenetic Reader Domain | Chromatin/Epigenetic |
IACS-9571 Hydrochloride is a selective and potent inhibitor of TRIM24 and BRPF1, (IC50: 8 nM for TRIM24; Kds: 31 nM and 14 nM for TRIM24 and BRPF1). |