Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20000 |
I-XW-053
4-(4,5-二苯基-1H-咪唑-2-基)苯甲酸 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
I-XW-053 是一种针对衣壳的 HIV-1 复制抑制剂,使用基于混合结构的方法以微摩尔亲和力阻断 CA N 末端结构域之间的界面(NTD-NTD 界面)。 | |||
T27642 |
I-XW-053 sodium
I-XW-053 Na,I XW 053 sodium,IXW053 sodium,I XW 053 Na,IXW053 Na |
||
I-XW-053 sodium inhibits the replication of a diverse panel of primary HIV-1 isolates in Peripheral blood mononuclear cell with no appreciable cytotoxicity. | |||
T27030 |
CK176
HIV-1 inhibitor-34,HIV-1 inhibitor 34,CK 176,CK-176,HIV-1 inhibitor34 |
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CK176 is a capsid targeted inhibitor of HIV-1 replication. CK176 shows an 11-fold improvement over I-XW-053 in blocking HIV-1 replication in primary human peripheral blood mononuclear cells (PBMCs). |