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Cat. No. Product Name Target Signaling Pathways
TP1900L1 Hemopressin (human, mouse) acetate

Hemopressin (human, mouse) acetate(1314035-51-2 free base)

Cannabinoid Receptor GPCR/G Protein
Hemopressin (human, mouse) acetate(1314035-51-2 free base) 是一种衍生自血红蛋白 α1 链的九肽,是从大鼠脑匀浆中分离出来的。 Hemopressin 是 CB1 大麻素受体的口服活性、选择性和反向激动剂。 Hemopressin 在炎性疼痛模型中发挥镇痛作用。
TP1901L1 Hemopressin (rat) acetate(568588-77-2 free base)

Cannabinoid Receptor GPCR/G Protein
Hemopressin (rat) acetate(568588-77-2 free base) 是一种衍生自血红蛋白 α1 链的九肽,起初是从大鼠脑匀浆中分离出来的。 Hemopressin 是 CB2 大麻素受体的口服活性、选择性和反向激动剂。 Hemopressin 在炎性疼痛模型中发挥镇痛作用。
TP1901 Hemopressin(rat)

Hemopressin (rat)

Bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE. Ki values are 27.76, 3.43 and 1.87 μM respectively. Potent hypotensive in vivo. Also acts as a selective CB1 receptor inverse agonist. Displays antinoc
TP1900 Hemopressin (human, mouse)

Bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE. Ki values are 27.76, 3.43 and 1.87 μM respectively. Potent hypotensive in vivo. Also acts as a selective CB1 receptor inverse agonist. Displays antinoc
T75798 Hemopressin(rat) TFA

Hemopressin(rat) TFA,一种衍生自α1-珠蛋白九肽,最初分离自大鼠脑匀浆。该化合物通过口服能有效选择性地作为CB1大麻素受体的反向激动剂,并在炎性疼痛模型中表现出抗伤害感受活性。
T75799 Hemopressin(human, mouse) TFA

Cannabinoid Receptor GPCR/G Protein
Hemopressin TFA,一种衍生自血红蛋白α1链的九肽,最初自大鼠脑匀浆分离。作为口服活性且选择性的CB1大麻素受体反向激动剂,Hemopressin TFA在炎性疼痛模型中具有抗伤害感受效应。
TP1939L1 RVD-Hpα acetate(1193362-76-3 free base)

Cannabinoid Receptor GPCR/G Protein
RVD-Hpα acetate(1193362-76-3 free base) 是人血加压素的 N 末端延伸形式,可作为选择性 CB1 受体激动剂。增加体外表达 CB1 受体的细胞中的细胞内 Ca2+ 水平。也是高亲和力 CB2 正变构调节剂 (Ki = 50 nM)。
T75936 RVD-Hpα TFA

RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selectiveCB1receptoragonist. RVD-Hpα TFA increases intracellular Ca2+levels in cells expressingCB1receptors in vitro. RVD-Hpα TFA also high affinityCB2positive allosteric modulator (Ki=50 nM).
TP1939 RVD-Hpα

N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM).

化合物

Hemopressin (human, mouse) acetate
Cat.No: TP1900L1
Synonym: Hemopressin (human, mouse) acetate(1314035-51-2 free base)
Target: Cannabinoid Receptor
Hemopressin (rat) acetate(568588-77-2 free base)
Cat.No: TP1901L1
Synonym:
Target: Cannabinoid Receptor
Hemopressin(rat)
Cat.No: TP1901
Synonym: Hemopressin (rat)
Target:
Hemopressin (human, mouse)
Cat.No: TP1900
Synonym:
Target:
Hemopressin(rat) TFA
Cat.No: T75798
Synonym:
Target:
Hemopressin(human, mouse) TFA
Cat.No: T75799
Synonym:
Target: Cannabinoid Receptor
RVD-Hpα acetate(1193362-76-3 free base)
Cat.No: TP1939L1
Synonym:
Target: Cannabinoid Receptor
RVD-Hpα TFA
Cat.No: T75936
Synonym:
Target:
RVD-Hpα
Cat.No: TP1939
Synonym:
Target:
TargetMol Loading
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