Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T82165 |
HTH-02-006
|
AMPK | Chromatin/Epigenetic; PI3K/Akt/mTOR signaling |
HTH-02-006,一种NUAK2抑制剂(IC50 = 126 nM),能够降低HuCCT-1细胞中磷酸化MYPT1水平,并抑制YAP驱动的细胞增殖、肝肿大和肿瘤发生,同时具备抗纤维化保护效果。 |