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18

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T17842	DOTA-NHS-ester	Others	Others
	DOTA-NHS-ester 是 affibody 分子的接头，应用于小动物 PET、SPECT 和 CT。它可用于标记放射治疗剂或成像探针以检测肿瘤。
T35447	10(S)-PAHSA
	10(S)-PAHSA is a stereoisomer of 10-PAHSA , an endogenous lipid that belongs to a collection of branched fatty acid esters of hydroxy fatty acids (FAHFAs).
T36588	9(R)-PAHSA
	9(R)-PAHSA is a stereoisomer of 9-PAHSA , an endogenous lipid that belongs to a collection of branched fatty acid esters of hydroxy fatty acids (FAHFAs).
T36586	12-PAHSA
	Branched fatty acid esters of hydroxy fatty acids (FAHFAs) are newly identified endogenous lipids regulated by fasting and high-fat feeding and associated with insulin sensitivity. Structurally, these esters are comprised of a C-16 or C-18 fatty acid (e.g., palmitoleic, palmitic, oleic, or stearic acid) linked to either a C-16 or C-18 hydroxy substituent. 12-PAHSA is a FAHFA in which palmitic acid is esterified at the 12th carbon of hydroxy stearic acid. Among the FAHFA family members, PAHSAs ar...
T35446	10(R)-PAHSA
	10(R)-PAHSA is a stereoisomer of 10-PAHSA , an endogenous lipid that belongs to a collection of branched fatty acid esters of hydroxy fatty acids (FAHFAs).
T36142	10-PAHSA
	10-PAHSA is a newly identified endogenous lipid that belongs to a collection of branched fatty acid esters of hydroxy fatty acids (FAHFAs). It is a FAHFA in which palmitic acid is esterified to 10-hydroxy stearic acid. Among the FAHFA family members, PAHSAs are the most abundant in the adipose tissue of glucose tolerant AG4OX mice, which overexpress the Glut4 glucose transporter specifically in adipose tissue. As other FAHFAs improve glucose tolerance, stimulate insulin secretion, and have anti-...
T36590	9-PAHSA
	Branched fatty acid esters of hydroxy fatty acids (FAHFAs) are newly identified endogenous lipids regulated by fasting and high-fat feeding and associated with insulin sensitivity. Structurally, these esters are comprised of a C-16 or C-18 fatty acid (e.g., palmitoleic, palmitic, oleic, or stearic acid) linked to a hydroxylated C-16 or C-18 lipid. 9-PAHSA is a FAHFA in which palmitic acid is esterified to 9-hydroxy stearic acid. PAHSAs are the most abundant forms of FAHFA in serum as well as whi...
T77724	OBHSA Oxabicycloheptane sulfonamide	Estrogen/progestogen Receptor	Endocrinology/Hormones
	OBHSA（Oxabicycloheptane sulfonamide）是一种新型选择性雌激素受体降解剂（SERD），可用于研究乳腺癌。
T24573	Ovatodiolide
	Ovatodiolide is a broad anticancer agent that acts by upregulating hsa-miR-155, suppressing the BCR-ABL fusion gene, and dysregulating the PI3K/AKT/mTOR pathway.
T29837	Albumin blue 670 AB670,AB-670,AB 670
	Albumin blue 670, as an Albumin probe, can bind to HSA to form a fluorescent complex.
T77146	Regavirumab
	Regavirumab (MCA C23)为针对巨细胞病毒(CMV)、人血清白蛋白(HSA)及氨基乙酸的人源单克隆抗体。
T82606	Dazodalibep MEDI 4920,VIB 4920
	Dazodalibep（MEDI 4920; VIB 4920）为针对CD40LG/TNFSF5的单克隆抗体，其结构中融合了ALB/HSA。
T82600	DDAO-C6
	DDAO-C6为酯环酮衍生物，高度特异性荧光探针，专用于检测人血清白蛋白(HSA)。同时，DDAO-C6作为酶激活的近红外荧光探针，适用于通过肠道微生物内源性脂肪酶的活性变化进行目测（Ex/Em=600/658 nm）。
T36398	Paclitaxel octadecanedioate
	Paclitaxel octadecanedioate is a prodrug form of paclitaxel that is comprised of paclitaxel conjugated to 1,18-octadecanedioic acid.1 Unlike paclitaxel, it does not promote tubulin polymerization in vitro when used at a concentration of 10 μM. A 5:1 mixture of paclitaxel octadecanedioate:human serum albumin (HSA) is cytotoxic to HT-1080, PANC-1, and HT-29 cells (IC50s = 12, 2.48, and 8.62 nM, respectively). This mixture reduces tumor growth and increases survival in an HT-1080 mouse xenograft mo...
T77126	Ozoralizumab
	Ozoralizumab (ATN-103) 为一种针对TNFα的人源化抗体。该化合物为一种三价人源化纳米抗体，由两个针对人TNFα的纳米抗体和一个针对人血清白蛋白(HSA)的纳米抗体构成，适用于关节炎研究。
T79282	Antibacterial agent 144
	Antibacterialagent 144（compound 8e）是一款效能超过氯霉素和阿莫西林的抗菌药物，专门针对具有多重耐药性的金黄色葡萄球菌。该化合物通过破坏细菌的细胞质膜和抑制生物膜形成来发挥作用。Antibacterialagent 144能与HSA紧密结合（Kd=13.2 μM），显示出卓越的杀菌活性。它还能与DNA相结合，形成超分子复合物，有效阻断DNA复制过程。
T83922	Pep2 Peptide
	Pep2 peptide是一种针对跨膜糖蛋白CD36的肽配体，CD36也被称为清道夫受体B2。在1 mM浓度使用时，Pep2 peptide在无细胞检测中选择性地与CD36结合，相比于人血清白蛋白(HSA)、IgG和CD44具有更高的亲和力。与不含Pep2 peptide的胶束相比，包裹抗癌剂多柔比星的Pep2 peptide功能化胶束能增加多柔比星在过表达CD36的HepG2肝细胞癌细胞中的细胞内输送，并提升细胞毒性。
T36713	Streptochlorin
	Streptochlorin is a bacterial metabolite originally isolated from Streptomyces sp. SF2583 that has diverse biological activities, including antiangiogenic, antiproliferative, and anti-allergic properties. It inhibits TNF-α-induced NF-κB transcriptional activity and decreases proliferation of human umbilical vein endothelial cells (HUVECs) when used at concentrations ranging from 5 to 20 μM. Streptochlorin (12 μg/ml) decreases viability of, as well as induces apoptosis and increases the productio...

化合物

Cat.No: T17842

Target: Others

Cat.No: T35447

Cat.No: T36588

Cat.No: T36586

Cat.No: T35446

Cat.No: T36142

Cat.No: T36590

Cat.No: T77724

Synonym: Oxabicycloheptane sulfonamide

Target: Estrogen/progestogen Receptor

Cat.No: T24573

Albumin blue 670

Cat.No: T29837

Synonym: AB670,AB-670,AB 670

Cat.No: T77146

Cat.No: T82606

Synonym: MEDI 4920,VIB 4920

Cat.No: T82600

Paclitaxel octadecanedioate

Cat.No: T36398

Cat.No: T77126

Antibacterial agent 144

Cat.No: T79282

Cat.No: T83922

Cat.No: T36713

Cat. No.	Product Name	Target	Signaling Pathways
TN1518	Cochinchinenin C	Others	Others
	There is a synergistic interaction between loureirin A and Cochinchinenin C, and the fluorescence quenching of HSA by loureirin A (or Cochinchinenin C) is a combined quenching procedure (dynamic and static quenching).
T83319	4-epi-Withaferin A
	4-epi-Withaferin A（化合物28）是Withaferin A的一个类似物，它增强了细胞毒性及细胞保护性热休克诱导活性（HSA）。此外，4-epi-Withaferin A还展现了通过激活细胞防御机制来研究蛋白质聚集相关疾病的潜力。

天然产物

Cochinchinenin C

Cat.No: TN1518

Target: Others

4-epi-Withaferin A

Cat.No: T83319

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