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Cat. No. Product Name Target Signaling Pathways
T16807 Rucaparib monocamsylate

瑞卡帕布樟脑磺酸盐,Rucaparib Camsylate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Rucaparib monocamsylate (Rucaparib Camsylate) 是一种口服有效的 PARP 蛋白抑制剂,对 PARP-1 的Ki 为 1.4 nM。它是六磷酸己糖脱氢酶 (H6PD) 抑制剂,有用于去势抵抗性前列腺癌 (CRPC) 的研究潜力。
T4463 Rucaparib

AG-14447,PF-01367338,瑞卡帕布,AG014699

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Rucaparib (PF-01367338) 是一种口服有效的 PARP 蛋白抑制剂,对 PARP-1 的 Ki 为 1.4 nM。它是六磷酸己糖脱氢酶 (H6PD) 抑制剂,有用于去势抵抗性前列腺癌 (CRPC) 的研究潜力。
T6127 Rucaparib Phosphate

AG-014699 phosphate,PF-01367338,芦卡帕利,AG-014699,瑞卡帕布磷酸盐,PF-01367338 phosphate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Rucaparib Phosphate (PF-01367338 phosphate) 是一种口服有效的PARP 蛋白抑制剂,对 PARP-1 的Ki 为 1.4 nM。它是六磷酸己糖脱氢酶 (H6PD) 抑制剂,有用于去势抵抗性前列腺癌 (CRPC) 的研究潜力。
T64289 Rucaparib camsylate

Rucaparib (AG014699) camsylate 是一种口服具有活力的 PARP 蛋白 (PARP-1、PARP-2 及 PARP-3) 抑制剂,对 PARP-1 的 Ki=1.4 nM。Rucaparib camsylate 是一种六磷酸己糖脱氢酶 (H6PD) 抑制剂。Rucaparib camsylate 具有潜力进行去势抵抗性前列腺癌 (CRPC) 的研究研究。
T63065 Rucaparib tartrate

Rucaparib (AG014699) tartrate 是一种口服具有活力的 PARP 蛋白 (PARP-1, PARP-2 和 PARP-3) 抑制剂,作用于 PARP-1 (Ki: 1.4 nM)。Rucaparib tartrate 是一种六磷酸己糖脱氢酶 (H6PD) 抑制剂。Rucaparib tartrate 具有潜力用于去势抵抗性前列腺癌 (CRPC) 的研究。
T61657 Rucaparib acetate

Rucaparib (AG014699) acetate is a highly effective oral inhibitor of PARP proteins, specifically targeting PARP-1, PARP-2, and PARP-3, with a Ki value of 1.4 nM for PARP1. Additionally, it exhibits inhibitory action on hexose-6-phosphate dehydrogenase (H6PD) to a moderate extent. Rucaparib acetate shows promise in the field of research for castration-resistant prostate cancer (CRPC). [1] [2] [3] [4]
T61335 Rucaparib hydrochloride

Rucaparib hydrochloride, also known as AG014699, is a powerful and orally active compound that inhibits PARP proteins including PARP-1, PARP-2, and PARP-3 with a Ki value of 1.4 nM for PARP1. Additionally, Rucaparib hydrochloride acts as a modest inhibitor of hexose-6-phosphate dehydrogenase (H6PD). This compound shows potential in research for castration-resistant prostate cancer (CRPC) [1] [2] [3] [4].

化合物

Rucaparib monocamsylate
Cat.No: T16807
Synonym: 瑞卡帕布樟脑磺酸盐,Rucaparib Camsylate
Target: PARP
Rucaparib
Cat.No: T4463
Synonym: AG-14447,PF-01367338,瑞卡帕布,AG014699
Target: PARP
Rucaparib Phosphate
Cat.No: T6127
Synonym: AG-014699 phosphate,PF-01367338,芦卡帕利,AG-014699,瑞卡帕布磷酸盐,PF-01367338 phosphate
Target: PARP
Rucaparib camsylate
Cat.No: T64289
Synonym:
Target:
Rucaparib tartrate
Cat.No: T63065
Synonym:
Target:
Rucaparib acetate
Cat.No: T61657
Synonym:
Target:
Rucaparib hydrochloride
Cat.No: T61335
Synonym:
Target:
TargetMol Loading
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