Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2770 |
Gentiopicroside
Gentiopicrin,龙胆苦甙,龙胆苦苷 |
P450; HCV Protease | Metabolism; Microbiology/Virology; Proteases/Proteasome |
Gentiopicroside (Gentiopicrin) 是天然环烯醚萜苷,具有抗炎和抗氧化活性。它抑制P450的活性,对 CYP2A6 的 IC50和 Ki 值分别为 61 µM 和 22.8 µM, | |||
T4S1439 |
6'-O-beta-D-Glucosylgentiopicroside
6'-O-β-D-葡萄糖基龙胆苦苷,6'-O-Glucosylgentiopicroside |
Antifungal | Microbiology/Virology |
6'-O-beta-D-Glucosylgentiopicroside (6'-O-Glucosylgentiopicroside) 是一种环烯醚萜,分离自G. straminea 根中。它能显著抑制 fMLP 诱导的超氧化物生成。 |