Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T27503 |
GV150013
GV 150013,GV-150013 |
cholecystokinin | GPCR/G Protein |
GV150013是一种 cholecystokinin-2 (CCK2)受体拮抗剂。 | |||
T27503L |
GV-150013X
(S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea |
cholecystokinin | GPCR/G Protein |
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) 是一种有效的CCKB 拮抗剂,pKi= 9.02。 |