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Cat. No. Product Name Target Signaling Pathways
T9573 GSK3685032

DNA Methyltransferase Chromatin/Epigenetic
GSK-3685032 是一种非时间依赖、非共价、选择性的、可逆的DNMT1抑制剂,IC50=0.036 μM。它诱导 DNA 甲基化丧失、转录激活和癌细胞生长抑制。
T39648 (R)-GSK-3685032

(R)-GSK-3685032 is the R-enantiomer of GSK-3685032. GSK-3685032 is a first-in-class, non-time-dependent, non-covalent, reversible, selective DNMT1 inhibitor with an IC 50 of 0.036 μM. GSK-3685032 induces robust loss of DNA methylation, transcriptional activation and inhibition of cancer cell growth.

化合物

GSK3685032
Cat.No: T9573
Synonym:
Target: DNA Methyltransferase
(R)-GSK-3685032
Cat.No: T39648
Synonym:
Target:
TargetMol Loading
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