Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15419 |
GS-626510
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2). |