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Cat. No. | Product Name | Target | Signaling Pathways |
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T36635 |
[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)
[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human) |
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[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human) 是GRF的 类似物,是一种血管活性肠肽 (VIP) 拮抗剂。 | |||
T83549 |
(D-Ala2)-GRF (1-29) amide (human)
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'(D-Ala2)-GRF (1-29) amide (human)' 为一种GRF的超激动剂,其GH释放活性在猪和大鼠体内极为显著,大约为GRF (1-29)活性的50倍。 | |||
T78039 |
Acetyl-(D-Arg2)-GRF (1-29) amide (human)
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Acetyl-(D-Arg2)-GRF (1-29) amide (human) 是一种针对人体的生长激素释放因子(GRF)拮抗剂,其主要作用是抑制生长激素(GH)的释放,广泛应用于内分泌学领域的研究。 | |||
T83491 |
[K15,R16,L27]VIP(1-7)/GRF(8-27)
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[K15,R16,L27]VIP(1-7)/GRF(8-27)作为VIP1激动剂,对人类VIP1、大鼠VIP1及大鼠VIP2的结合IC50分别为2 nM、1 nM和30000 nM。 | |||
T78035 |
[K15,R16,L27]VIP(1-7)/GRF(8-27) acetate
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[K15,R16,L27]VIP(1-7)/GRF(8-27)(acetate)为[K15,R16,L27]VIP(1-7)/GRF(8-27)的醋酸盐形态,作为VIP1激动剂,与人类和大鼠的肠血管活性肽1 (VIP 1) 及大鼠的肠血管活性肽2 (VIP 2) 的结合IC50值分别为2 nM、1 nM和30000 nM。 | |||
T83195 |
Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
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Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27),是一种血管活性肠肽,起到VIP1受体拮抗剂的作用。 | |||
TP2328L |
CJC-1295 acetate(863288-34-0 free base)
DAC:GRF acetate |
GHSR | GPCR/G Protein |
CJC-1295 acetate(863288-34-0 free base) (DAC:GRF acetate) 是生长激素释放激素 (GHRH)(也称为生长激素释放因子 (GRF))和生长激素促分泌素 (GHS) 的合成类似物。 | |||
TP2103 |
[D-p-Cl-Phe6,Leu17]-VIP
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Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors. | |||
T78003 |
[D-p-Cl-Phe6,Leu17]-VIP TFA
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[D-p-Cl-Phe6,Leu17]-VIP TFA,为竞争性及选择性血管活性肠肽(VIP)受体拮抗剂,其IC50为125.8 nM。该化合物针对胰高血糖素、促胰液素和GRF受体均不表现活性。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-00186 |
GHRH Protein, Human, Recombinant (hFc)
GRF,INN,growth hormone releasing hormone,GHRF |
Human | HEK293 Cells |
The role of hypothalamic growth hormone-releasing hormone (GHRH) in the release of growth hormone (GH) from the pituitary is well established. Extra-hypothalamic growth hormone-releasing hormone (GHRH) plays an important role in infertility. Growth hormone releasing hormone (GHRH) has recently been shown to increase the level of gamma-aminobutyric acid (GABA) and activate GABA receptors (GABARs) in the cerebral cortex. GABA is an inhibitory neurotransmitter that can inhibit seizures. GHRH may pl... |