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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T36635 [Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)

[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)

[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human) 是GRF的 类似物,是一种血管活性肠肽 (VIP) 拮抗剂。
T83549 (D-Ala2)-GRF (1-29) amide (human)

'(D-Ala2)-GRF (1-29) amide (human)' 为一种GRF的超激动剂,其GH释放活性在猪和大鼠体内极为显著,大约为GRF (1-29)活性的50倍。
T78039 Acetyl-(D-Arg2)-GRF (1-29) amide (human)

Acetyl-(D-Arg2)-GRF (1-29) amide (human) 是一种针对人体的生长激素释放因子(GRF)拮抗剂,其主要作用是抑制生长激素(GH)的释放,广泛应用于内分泌学领域的研究。
T83491 [K15,R16,L27]VIP(1-7)/GRF(8-27)

[K15,R16,L27]VIP(1-7)/GRF(8-27)作为VIP1激动剂,对人类VIP1、大鼠VIP1及大鼠VIP2的结合IC50分别为2 nM、1 nM和30000 nM。
T78035 [K15,R16,L27]VIP(1-7)/GRF(8-27) acetate

[K15,R16,L27]VIP(1-7)/GRF(8-27)(acetate)为[K15,R16,L27]VIP(1-7)/GRF(8-27)的醋酸盐形态,作为VIP1激动剂,与人类和大鼠的肠血管活性肽1 (VIP 1) 及大鼠的肠血管活性肽2 (VIP 2) 的结合IC50值分别为2 nM、1 nM和30000 nM。
T83195 Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)

Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27),是一种血管活性肠肽,起到VIP1受体拮抗剂的作用。
TP2328L CJC-1295 acetate(863288-34-0 free base)

DAC:GRF acetate

GHSR GPCR/G Protein
CJC-1295 acetate(863288-34-0 free base) (DAC:GRF acetate) 是生长激素释放激素 (GHRH)(也称为生长激素释放因子 (GRF))和生长激素促分泌素 (GHS) 的合成类似物。
TP2103 [D-p-Cl-Phe6,Leu17]-VIP

Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.
T78003 [D-p-Cl-Phe6,Leu17]-VIP TFA

[D-p-Cl-Phe6,Leu17]-VIP TFA,为竞争性及选择性血管活性肠肽(VIP)受体拮抗剂,其IC50为125.8 nM。该化合物针对胰高血糖素、促胰液素和GRF受体均不表现活性。

化合物

[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)
Cat.No: T36635
Synonym: [Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)
Target:
(D-Ala2)-GRF (1-29) amide (human)
Cat.No: T83549
Synonym:
Target:
Acetyl-(D-Arg2)-GRF (1-29) amide (human)
Cat.No: T78039
Synonym:
Target:
[K15,R16,L27]VIP(1-7)/GRF(8-27)
Cat.No: T83491
Synonym:
Target:
[K15,R16,L27]VIP(1-7)/GRF(8-27) acetate
Cat.No: T78035
Synonym:
Target:
Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
Cat.No: T83195
Synonym:
Target:
CJC-1295 acetate(863288-34-0 free base)
Cat.No: TP2328L
Synonym: DAC:GRF acetate
Target: GHSR
[D-p-Cl-Phe6,Leu17]-VIP
Cat.No: TP2103
Synonym:
Target:
[D-p-Cl-Phe6,Leu17]-VIP TFA
Cat.No: T78003
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-00186 GHRH Protein, Human, Recombinant (hFc)

GRF,INN,growth hormone releasing hormone,GHRF

Human HEK293 Cells
The role of hypothalamic growth hormone-releasing hormone (GHRH) in the release of growth hormone (GH) from the pituitary is well established. Extra-hypothalamic growth hormone-releasing hormone (GHRH) plays an important role in infertility. Growth hormone releasing hormone (GHRH) has recently been shown to increase the level of gamma-aminobutyric acid (GABA) and activate GABA receptors (GABARs) in the cerebral cortex. GABA is an inhibitory neurotransmitter that can inhibit seizures. GHRH may pl...

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GHRH Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00186
Species: Human
Expression System: HEK293 Cells
TargetMol Loading
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