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Cat. No. Product Name Target Signaling Pathways
T11452 GPR120 Agonist 1

GPR Endocrinology/Hormones; GPCR/G Protein
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively.
T15413 GPR120 Agonist 3

GPR120-IN-1

GPR Endocrinology/Hormones; GPCR/G Protein
GPR120 Agonist 3 (GPR120-IN-1) 是一种有效的、选择性的 Gpr120激动剂,logEC50为 −7.62。
T22967 MEDICA16

MEDICA 16

GPR; Others; ATP Citrate Lyase Endocrinology/Hormones; GPCR/G Protein; Metabolism; Others
MEDICA16 是 GPR40 的特异性激动剂以及 GPR120 的部分激动剂。 MEDICA16 是一种 ATP-柠檬酸裂解酶抑制剂,可显着降低腓肠肌中的细胞内 TG 含量,同时增加胰岛素敏感性。
T28140 NCG21

NCG-21,NCG 21

NCG21 is a GPR120 agonist, which showed potent extracellular signal-regulated kinase (ERK) activation in a cloned GPR120 system. NCG21 potently activated ERK, intracellular calcium responses and GLP-1 secretion in murine enteroendocrine STC-1 cells that e

化合物

GPR120 Agonist 1
Cat.No: T11452
Synonym:
Target: GPR
GPR120 Agonist 3
Cat.No: T15413
Synonym: GPR120-IN-1
Target: GPR
MEDICA16
Cat.No: T22967
Synonym: MEDICA 16
Target: GPR, Others, ATP Citrate Lyase
NCG21
Cat.No: T28140
Synonym: NCG-21,NCG 21
Target:
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