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Cat. No. | Product Name | Target | Signaling Pathways |
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T68568 |
Encequidar, HCl
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Encequidar, also known as HM-30181, is an oral P-glycoprotein (P-gp) inhibitor developed to enhance the oral bioavailability of P-gp substrate drugs. Encequidar showed the highest potency (IC(50)=0.63nM) among several MDR1 inhibitors, including cycloporin A, XR9576, and GF120918, and effectively blocked transepithelial transport of paclitaxel in MDCK monolayers (IC(50)=35.4nM). Encequidar is currently under clinical trials. | |||
T72678 |
P-gp inhibitor 4
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P-gp inhibitor 4 是一种选择性的 P-glycoprotein 调节剂,EC50值为 94 nM。P-gp inhibitor 4 增加药物通过胃肠道屏障的能力,恢复 doxorubicin 在耐药癌细胞中的毒性。 | |||
T75766 |
GP(33-41) TFA
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GP(33-41) TFA 是一种由 9 个氨基酸残基组成的多肽,它是淋巴细胞性脉络丛脑膜炎病毒 GP1 抗原决定基中的序列。GP(33-41) TFA 能够上调 RMA-S (Db Kb) 细胞表面 H-2Db 分子,SC50值为 344 nM。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-01262 |
TROP-2 Protein, Human, Recombinant (His)
TROP2,M1S1,GA733-1,TROP-2,GA7331,tumor-associated calcium si... |
Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.4 kDa and the accession number is P09758. | |||
TMPY-06972 |
TROP-2 Protein, Human, Recombinant (hFc)
EGP-1,GA733-1,tumor-associated calcium signal trans... |
Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 54.6 kDa and the accession number is NP_002344.2. | |||
TMPY-00946 |
TROP-2 Protein, Human, Recombinant (His & hFc)
GP50,TACD2,GA733-1,M1S1,GA7331,EGP |
Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 55.7 kDa and the accession number is P09758. | |||
TMPY-06378 |
TROP-2 Protein, Human, Recombinant (His & Avi), Biotinylated
EGP-1,GA733-1,GP50,TACD2,TROP2,E<... |
Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 31.14 kDa and the accession number is NP_002344.2. | |||
TMPY-06720 |
TROP-2 Protein, Human, Recombinant (hFc & Avi), Biotinylated
GA733-1,EGP1,GP50,TROP-2,GA7331,E... |
Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 56.42 kDa and the accession number is NP_002344.2. |