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Cat. No.	Product Name	Target	Signaling Pathways
T4664	ML 297 ML297	Potassium Channel	Membrane transporter/Ion channel
	ML 297 是选择性的 GIRK1/2激活剂，EC50为 0.16 μM。ML 297 在癫痫病的研究中具有价值。
T7899	VU0810464	Potassium Channel	Membrane transporter/Ion channel
	VU0810464 是一种选择性的非尿素蛋白门控的内向整流钾通道激活剂。 VU0810464对神经元 GIRK1/2和GIRK1/4 的EC50分别为165 nM 和720 nM。VU0810464具有脑部渗透性。
T17246	VU0529331	Others	Others
	VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel activator (EC50s: 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively). It is also effective on the GIRK4 homomeric channel.
T27502	Gue1654 Gue-1654,Gue 1654
	Gue1654 is a modulator of oxoeicosanoid receptor 1 (OXE-R). Gue1654 selectively inhibits Gβγ upon activation of the Gαi-βγ heterotrimer by OXE-R. Gue1654 inhibits Gβγ-mediated opening of GIRK1/2 channels in HEK293 cells.