Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78104 |
Fosnetupitant chloride monohydrochloride
Pronetupitant chloride monohydrochloride |
Neurokinin receptor | GPCR/G Protein; Neuroscience |
Fosnetupitant chloride monohydrochloride(Pronetupitant chloride monohydrochloride)为NK1受体拮抗剂,对人NK1受体和NK3受体的pKi分别为9.5和6.1。它是奈妥匹坦的亚甲基磷酸酯前体。 |