Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T39808 |
Firazorexton
|
||
Firazorexton is a potent orexin type 2 receptor (OX2R) agonist. | |||
T78636 |
Firazorexton hydrate
TAK-994 |
||
Firazorexton hydrate (TAK-994)为一种高效的食欲素2型受体(OX2R)激动剂,EC50值为19 nM。在发作性睡病小鼠模型中,该化合物能够有效减少觉醒碎片和猝倒样发作的发生。 |