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Cat. No. Product Name Target Signaling Pathways
T15275 Fenobam

GluR Neuroscience
Fenobam 是可口服的、可穿过血脑屏障的 mGluR5拮抗剂,具有抗焦虑活性,在大鼠和人重组 mGlu5 受体上的 Kd 值分别 54 和 31 nM。它有反向激动剂活性,可阻断 mGlu5 受体活性,IC50为 84 nM。
T68959 Fenobam hydrate

Fenobam hydrate is a noncompetitive antagonist and inverse agonist of metabotropic glutamate receptor 5 (mGluR5). It inhibits intracellular calcium mobilization induced by the glutamate analog quisqualate and inhibits basal activity of mGluR5. Fenobam reduces stress-induced hyperthermia, exhibits anxiolytic-like activity, and may induce analgesia.

化合物

Fenobam
Cat.No: T15275
Synonym:
Target: GluR
Fenobam hydrate
Cat.No: T68959
Synonym:
Target:
TargetMol Loading
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