Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1263 |
Fz7-21
(Ac)-LPSDDLEFWCHVMY-NH2 |
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
Fz7-21 ((Ac)-LPSDDLEFWCHVMY-NH2) 是一种 Frizzled 7 (FZD 7) 受体的肽抑制剂,能够选择性的与FZD7 CRD 亚类结合。它还阻断了WNT3A 介导的β-catenin 在小鼠L 细胞中的稳定作用。它对外源性WNT3A 刺激和转染WNT3A 或WNT1的HEK293细胞Wnt/β-catenin 信号传导有损伤。 | |||
T77692 |
F7H
|
Wnt/beta-catenin; Antibacterial | Cytoskeletal Signaling; Microbiology/Virology; Stem Cells |
F7H 是一种有效的卷曲蛋白受体 (Frizzled receptor) FZD7 拮抗剂,IC50 值为 1.25 μM。F7H 是一种有效的 FZD7 跨膜结构域 (TMD) 的配体,具有潜在的抗肿瘤和抑菌活性。 | |||
T9662 |
SRI 37892
|
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
SRI 37892是一种 Fzd7抑制剂,对 Wnt/β-catenin 信号传导和癌症细胞活性具有强大的活性。 | |||
T75956 |
Fz7-21 TFA
|
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Fz7-21 (Ac-LPSDDLEFWCHVMY-NH2) TFA 是一种有效的 FZD7受体的肽拮抗剂,选择性地结合到 FZD7 CRD 亚类,并改变 CRD 的构象及其脂质结合槽的结构。人和小鼠 FZD7 CRD 的 EC50值分别为 58 和 34 nM。Fz7-21 TFA 损害 FZD7 在 Wnt-β-catenin 信号传导中的功能和肠类器官中的干细胞功能。 | |||
TP1262 |
Fz7-21 TFA (2247635-23-8 free base)
Fz7-21 TFA,(Ac)-LPSDDLEFWCHVMY-NH2 TFA |
||
Fz7-21 TFA ((Ac)-LPSDDLEFWCHVMY-NH2 TFA), a peptide antagonist of Frizzled 7 (FZD 7) receptors, selectively binds to FZD7 CRD subclass. The EC50 values are 58 and 34 nM for human and mouse FZD7 CRD, respectively. | |||
T68468 |
FJ9
|
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FJ9 is a FZD7 inhibitor which disrupts protein-protein interaction between Frz7 and the PDZ domain of DVL, and induces apoptosis in melanoma cell line and non-small cell lung cancer cell line. |