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Cat. No. Product Name Target Signaling Pathways
T11309 FMF-04-159-2

CDK Cell Cycle/Checkpoint
FMF-04-159-2 inhibits CDK14 and CDK2 with IC50s of 39.6 nM and 256 nM in NanoBRET assay, respectively. FMF-04-159-2 is a covalent CDK14 inhibitor.
T36305 FMF-04-159-R

Potent inhibitor of CDK16 and CDK14 (IC50 values are 6 and 140 nM, respectively in kinase activity assay; IC50 = 563 nM for CDK14 in BRET assay). Also binds CDK2 (IC50 = 493 nM). Inhibition reversible upon compound wash-out. Control for FMF-04-159-2 (Cat. No. 7158).

化合物

FMF-04-159-2
Cat.No: T11309
Synonym:
Target: CDK
FMF-04-159-R
Cat.No: T36305
Synonym:
Target:
TargetMol Loading
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