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Cat. No. Product Name Target Signaling Pathways
T79688 FAK-IN-11

FAK Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
FAK-IN-11 (Compound 4l) 作为FAK抑制剂,与FAK的ATP结合袋相结合,进而抑制其蛋白磷酸化。该化合物对MDA-MB-231细胞具有细胞毒性,IC50值为 13.73μM,并能诱导该细胞通过非凋亡途径死亡。
T41164 FC 11

FC 11 is a highly potent focal adhesion Ki nase (FAK) PROTAC®Degrader (DC50 values are 40 to 370 pM depending on cell line), which is composed of the FAK inhibitor PF 562217 joined by a linker to the cereblon-binding ligand Pomalidomide. The effects of FC 11 are reversible upon compound wash out. FC 11 also degrades autophosphorylated FAK (pFAKtyr397), displaying near complete degradation after 3 hours at 100 nM in TM3 cells.

化合物

FAK-IN-11
Cat.No: T79688
Synonym:
Target: FAK
FC 11
Cat.No: T41164
Synonym:
Target:
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