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Cat. No.	Product Name	Target	Signaling Pathways
T3179	Eptapirone F 11440	5-HT Receptor	GPCR/G Protein; Neuroscience
	Eptapirone (F 11440) 是一种高效且选择性的 5-HT1A 受体激动剂，具有显着的抗抑郁和抗焦虑潜力。
T71916	GSK-J1 sodium salt
	GSK-J1 sodium salt is a potent inhibitor of the H3K27 histone demethylases JMJD3 and UTX.
T70183	Eptapirone fumarate
	Eptapirone, also known as F11440, is a potent 5HT(1A) receptor agonist with marked anxiolytic and antidepressant potential. The affinity of F 11440 for 5-HT1A binding sites (pKi, 8.33) was higher than that of buspirone (pKi, 7.50), and somewhat lower than that of flesinoxan (pKi, 8.91). In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone, in exerting 5-HT1A agonist activity at pre- and postsynaptic receptors in rats (measured by, for exam...