Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T39497 |
EZH2-IN-4
EZH2-IN-4 |
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EZH2-IN-4 is a highly potent EZH2 inhibitor that can be taken orally. It exhibits inhibitory effects against wild type (WT) 5-membered (5-mer) EZH2 and mutant 5-mer EZH2, with IC 50 values of 0.923 nM and 2.65 nM, respectively. Moreover, EZH2-IN-4 has demonstrated significant anti-cancer activity. |