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Cat. No. Product Name Target Signaling Pathways
T4061 LY2334737

Nucleoside Antimetabolite/Analog; Others; Virus Protease Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
LY2334737 是一种具有口服活性的 Gemcitabine 的前药,也是核苷类似物。它抑制肠道病毒 A71 感染,有抗病毒和抗癌活性。
T61462 EV-A71-IN-1

EV-A71-IN-1 is a potent inhibitor of the human enterovirus A71 (EV-A71) capsid protein, with an EC50 of 0.27 μM against EV-A71. Acting as a capsid binder, EV-A71-IN-1 disrupts the crucial interaction between the viral VP1 protein and the host receptor hSCARB2. It displays broad-spectrum antiviral activity against various human enteroviruses, while being non-toxic to human cells (CC50 > 56.2 μM) [1].
T74487 AL-470

AL-470 是一个有效的抗病毒剂,对HIV-1、HIV-2、EV-A71的EC50值分别为0.27、0.63 和 0.35 µM。
T60880 Viral 2C protein inhibitor 1

Viral 2C protein inhibitor 1 (compound 6aw) 是广谱抗肠病毒剂,可抑制病毒 2C 蛋白。Viral 2C protein inhibitor 1 具有相对较低的细胞毒性和较高的选择性指数。Viral 2C protein inhibitor 1 可抑制 EV-D68、EV-A71 和 CVB3 等多种菌株,EC50值为 0.1~3.6 μM。

化合物

LY2334737
Cat.No: T4061
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Virus Protease
EV-A71-IN-1
Cat.No: T61462
Synonym:
Target:
AL-470
Cat.No: T74487
Synonym:
Target:
Viral 2C protein inhibitor 1
Cat.No: T60880
Synonym:
Target:
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