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Cat. No. Product Name Target Signaling Pathways
T11167 EHMT2-IN-2

Others Others
EHMT2-IN-2 Used in the research of blood disease or cancer. EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2.
T11166 EHMT2-IN-1

Others Others
EHMT2-IN-1 is a potent EHMT inhibitor, . Used in the research of blood disorder or cancer.with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2.
T7378 BRD9539

Histone Methyltransferase Chromatin/Epigenetic
BRD9539 是一种组蛋白甲基转移酶G9a 抑制剂,IC50为 6.3 μM,还抑制PRC2活性。
T1923 BRD4770

Histone Methyltransferase Chromatin/Epigenetic
BRD4770 是组蛋白甲基转移酶G9a 抑制剂,可激活共济失调毛细血管扩张突变途径并诱导细胞衰老。它可抑制H3K9的二甲基和三甲基化,EC50为 5 µM。
T60786 CSV0C018875

CSV0C018875 是基于喹啉的EHMT2/G9a 抑制剂,其细胞毒性低于 BIX-01294。
T71824 CSV0C018875 Hydrochloride

CSV0C018875 Hydrochloride is a novel G9a (EHMT2) inhibitor, binding tightly inside the active site cavity of G9a, inhibiting the activity of G9a in both enzyme and cell based assays with much lesser toxicity than BIX-0129.
T22250 5WKS

ZINC97756584

Others Others
5WKS 也称为ZINC97756584,是一种生物化学物质。它是G9a 蛋白抑制剂。G9A/EHMT2是一种核组蛋白赖氨酸甲基转移酶,催化H3K9me2,这是一种通常与转录基因沉默相关的可逆修饰。5WKS 可用于自身免疫性疾病或肿瘤的研究。

化合物

EHMT2-IN-2
Cat.No: T11167
Synonym:
Target: Others
EHMT2-IN-1
Cat.No: T11166
Synonym:
Target: Others
BRD9539
Cat.No: T7378
Synonym:
Target: Histone Methyltransferase
BRD4770
Cat.No: T1923
Synonym:
Target: Histone Methyltransferase
CSV0C018875
Cat.No: T60786
Synonym:
Target:
CSV0C018875 Hydrochloride
Cat.No: T71824
Synonym:
Target:
5WKS
Cat.No: T22250
Synonym: ZINC97756584
Target: Others
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