Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11158 |
EGFR-IN-11
|
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
EGFR-IN-11 是 EGFR-酪氨酸激酶的选择性抑制剂,可诱导细胞凋亡。 EGFR-IN-11 抑制三重突变体 EGFRL858R/T790M/C797S,IC50 为 18 nM,并在 G0/G1 时阻止细胞周期。 |