Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11081 | Dot1L-IN-1 | Histone Methyltransferase | Chromatin/Epigenetic |
The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor. | |||
T73637 | Dot1L-IN-1 TFA | ||
Dot1L-IN-1 TFA 是一种高效选择性Dot1L抑制剂,具有2 pM的Ki值和小于0.1 nM的IC50值。在HeLa细胞中,它能有效抑制H3K79的二甲基化(IC50=3 nM),同时也能在Molm-13细胞中抑制HoxA9启动子的活性(IC50=17 nM)。 |