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Cat. No. Product Name Target Signaling Pathways
T6476 Dofetilide

UK 68789,UK-68798,Tikosyn,多非利特

Potassium Channel Membrane transporter/Ion channel
Dofetilide (UK 68789) 是一种具有口服活性、有效的且特异性的IKr 阻滞剂,作为 III 类抗心律失常药物。Dofetilide 可用于心血管疾病研究。
T11072 Dofetilide D4

多非利特 D4,UK 68789 D4

Others Others
Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.
T11073 Dofetilide N-oxide

UK-116856

Others Others
Dofetilide N-oxide (UK-116856) is a metabolite of dofetilide. Dofetilide can block potassium channels and is a tertiary antiarrhythmic drug.
T16796 RPR-260243

Others Others
RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).

化合物

Dofetilide
Cat.No: T6476
Synonym: UK 68789,UK-68798,Tikosyn,多非利特
Target: Potassium Channel
Dofetilide D4
Cat.No: T11072
Synonym: 多非利特 D4,UK 68789 D4
Target: Others
Dofetilide N-oxide
Cat.No: T11073
Synonym: UK-116856
Target: Others
RPR-260243
Cat.No: T16796
Synonym:
Target: Others
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