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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20024 |
Tadalafil, (6R ,12aS)-
Tadalafil (6R ,12aS)- Lilly,Tadalafil specified impurity A,(-)-Tadalafil (6R ,12aS) diastereomer |
||
Tadalafil is a carboline derivative and Phosphodiesterase 5 Inhibitor. It is used primarily to treat Erectile dysfunction, Benign Prostatic Hyperplasia, and Primary Pulmonary Hypertension. | |||
T12961 |
Sofosbuvir impurity F
索非布韦杂质 F,Sofosbuvir 3',5'-Bis-(S)-phosphate |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) 既是 Sofosbuvir 的非对映异构体,也是 Sofosbuvir 的杂质,Sofosbuvir 是 HCV RNA 复制的抑制剂。 | |||
T12962 |
Sofosbuvir impurity G
|
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
Sofosbuvir impurity G 是 Sofosbuvir 的非对映异构体,是 Sofosbuvir 的杂质。其中 Sofosbuvir 能够抑制 HCVRNA 的复制,具有抗丙型肝炎病毒作用。 | |||
T74412 | dTAGV-1-NEG TFA | ||
dTAGV-1-NEG TFA 是一种非对映异构体,是 dTAGV-1 的异双功能阴性对照。dTAGV-1-NEG TFA 是一种 FKBP12F36V 选择性降解剂。 | |||
T38817 |
Golgicide A-1
GCA-1,Golgicide A-1 |
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Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction. | |||
T22356 | LLY-284 | Others | Others |
LLY-284 is the diastereomer of LLY-283, which is a selective and potent SAM-competitive chemical probe for PRMT5. LLY-284 is much less active than LLY-283 and can be used as a negative control for LLY-283. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13681 |
Epi-galantamine
|
AChE | Neuroscience |
Epi-galantamine 是 Galantamine 的非对映异构体,是从高加索雪花莲的鳞茎和花朵中分离出来的生物碱。它能够抑制AChE,EC50=45.7 μM 。 | |||
T7529 |
Yamogenin
山药 |
Others | Others |
Yamogenin 是一种薯蓣皂素的非对映异构体。它通过抑制 HepG2 肝细胞中脂肪酸合成的基因表达来抑制甘油三酸酯 (TG) 的积累。它在萤光素酶配体测定中拮抗肝脏 X 受体 (LXR) 的激活。 |