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6

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
T20024 Tadalafil, (6R ,12aS)-

Tadalafil (6R ,12aS)- Lilly,Tadalafil specified impurity A,(-)-Tadalafil (6R ,12aS) diastereomer

Tadalafil is a carboline derivative and Phosphodiesterase 5 Inhibitor. It is used primarily to treat Erectile dysfunction, Benign Prostatic Hyperplasia, and Primary Pulmonary Hypertension.
T12961 Sofosbuvir impurity F

索非布韦杂质 F,Sofosbuvir 3',5'-Bis-(S)-phosphate

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) 既是 Sofosbuvir 的非对映异构体,也是 Sofosbuvir 的杂质,Sofosbuvir 是 HCV RNA 复制的抑制剂。
T12962 Sofosbuvir impurity G

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sofosbuvir impurity G 是 Sofosbuvir 的非对映异构体,是 Sofosbuvir 的杂质。其中 Sofosbuvir 能够抑制 HCVRNA 的复制,具有抗丙型肝炎病毒作用。
T74412 dTAGV-1-NEG TFA

dTAGV-1-NEG TFA 是一种非对映异构体,是 dTAGV-1 的异双功能阴性对照。dTAGV-1-NEG TFA 是一种 FKBP12F36V 选择性降解剂。
T38817 Golgicide A-1

GCA-1,Golgicide A-1

Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction.
T22356 LLY-284

Others Others
LLY-284 is the diastereomer of LLY-283, which is a selective and potent SAM-competitive chemical probe for PRMT5. LLY-284 is much less active than LLY-283 and can be used as a negative control for LLY-283.

化合物

Tadalafil, (6R ,12aS)-
Cat.No: T20024
Synonym: Tadalafil (6R ,12aS)- Lilly,Tadalafil specified impurity A,(-)-Tadalafil (6R ,12aS) diastereomer
Target:
Sofosbuvir impurity F
Cat.No: T12961
Synonym: 索非布韦杂质 F,Sofosbuvir 3',5'-Bis-(S)-phosphate
Target: HCV Protease
Sofosbuvir impurity G
Cat.No: T12962
Synonym:
Target: HCV Protease
dTAGV-1-NEG TFA
Cat.No: T74412
Synonym:
Target:
Golgicide A-1
Cat.No: T38817
Synonym: GCA-1,Golgicide A-1
Target:
LLY-284
Cat.No: T22356
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T13681 Epi-galantamine

AChE Neuroscience
Epi-galantamine 是 Galantamine 的非对映异构体,是从高加索雪花莲的鳞茎和花朵中分离出来的生物碱。它能够抑制AChE,EC50=45.7 μM 。
T7529 Yamogenin

山药

Others Others
Yamogenin 是一种薯蓣皂素的非对映异构体。它通过抑制 HepG2 肝细胞中脂肪酸合成的基因表达来抑制甘油三酸酯 (TG) 的积累。它在萤光素酶配体测定中拮抗肝脏 X 受体 (LXR) 的激活。

天然产物

Epi-galantamine
Cat.No: T13681
Synonym:
Target: AChE
Yamogenin
Cat.No: T7529
Synonym: 山药
Target: Others
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