Cat. No. | Product Name | Target | Signaling Pathways |
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T7639 |
Deltorphin 2
Deltorphin 2(TFA),[D-Ala2]-Deltorphin II |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Deltorphin 2 ([D-Ala2]-Deltorphin II) 是一种选择性的 δ 阿片受体肽激动剂,IC50 为 1 nM。 | |||
T75770 |
Deltorphin 2 TFA
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Deltorphin 2 TFA 是一种选择性的 δ 阿片受体肽激动剂。 | |||
T36722 |
Deltorphin II (trifluoroacetate salt)
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Deltorphin II is a peptide agonist of δ2-opioid receptors.1,2It is selective for δ-opioid receptors over μ- and κ-opioid receptors in radioligand bindings assays (Kis = 0.0033, >1, and >1 μM, respectively) and induces [35S]GTPγS binding in mouse brain membrane preparations (EC50= 0.034 μM). Deltorphin II (0.12 mg/kg) decreases the infarction zone:risk zone ratio in a rat model of myocardial ischemia-reperfusion injury induced by coronary occlusion, an effect that can be reversed by the δ2-opioid... |