Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7637 |
Deltorphin I
Deltorphin 1,Deltorphin I(TFA),Deltorphin C |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Deltorphin I 是 δ-阿片受体的激动剂。 | |||
T36722 |
Deltorphin II (trifluoroacetate salt)
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Deltorphin II is a peptide agonist of δ2-opioid receptors.1,2It is selective for δ-opioid receptors over μ- and κ-opioid receptors in radioligand bindings assays (Kis = 0.0033, >1, and >1 μM, respectively) and induces [35S]GTPγS binding in mouse brain membrane preparations (EC50= 0.034 μM). Deltorphin II (0.12 mg/kg) decreases the infarction zone:risk zone ratio in a rat model of myocardial ischemia-reperfusion injury induced by coronary occlusion, an effect that can be reversed by the δ2-opioid... |