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Cat. No. Product Name Target Signaling Pathways
T16083 Mizagliflozin

GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base

SGLT GPCR/G Protein
Mizagliflozin (GSK-1614235 free base) 是口服有效的、选择性的 SGLT1抑制剂,对人 SGLT1 的 Ki 值为 27 nM。Mizagliflozin 对 SGLT1 的选择性是 SGLT2的303 倍。它是抗糖尿病药物,可以改善餐后血糖波动。它在改善慢性便秘方面具有潜在的作用。
T71340 Mizagliflozin sebacate

Mizagliflozin sebacate is a sodium-glucose transporter inhibitor. It is expected to improve postprandial hyperglycemia by suppressing glucose absorption from the intestine with a novel mechanism of action different from that of conventional alpha-glucosidase inhibitors. Mizagliflozin blocks intestinal glucose absorption and reduce GIP secretion in rats and humans, suggesting SGLT1 glucose transport is critical for GIP release.

化合物

Mizagliflozin
Cat.No: T16083
Synonym: GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base
Target: SGLT
Mizagliflozin sebacate
Cat.No: T71340
Synonym:
Target:
TargetMol Loading
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