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Cat. No. Product Name Target Signaling Pathways
T68566 Pitavastatin methyl ester

Pitavastatin methyl ester is the methyl ester derivative of Pitavastatin -- a competitive inhibitor of HMG-CoA reductase and an anti-lipemic agent.
T70077 Fadolmidine HCl

Fadolmidine, also known as MPV-2426, is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia. Fadolmidine displayed high affinity and full agonist efficacy at all three human alpha2-adrenoceptor subtypes (A, B and C) in transfected CHO cells with EC50 values (nM) of 0.4, 4.9 and 0.5, respectively. Fadolmidine inhibited also electrically evoked contractions in rat vas deferens demonstrating the activation of rodent presynaptic alpha2D-adrenoceptors with an ...
T70078 Fadolmidine

Fadolmidine is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia.

化合物

Pitavastatin methyl ester
Cat.No: T68566
Synonym:
Target:
Fadolmidine HCl
Cat.No: T70077
Synonym:
Target:
Fadolmidine
Cat.No: T70078
Synonym:
Target:
TargetMol Loading
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