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Cat. No. Product Name Target Signaling Pathways
T82595 DEALA-Hyp-YIPD

DEALA-Hyp-YIPD为HIF-1α抑制剂,阻断VHL/HIF-1α相互作用,显示IC50值为0.91 μM,Kd为180 nM。
T41172 FAM-DEALA-Hyp-YIPD

FAM-DEALA-Hyp-YIPD is a fluorescent HIF-1α peptide (Kd= 180-560 nM). Can be used to assess VHL binding in Fluorescence Polarization (FP) displacement assay, and evaluate the effect of VHL binding on degradation activity. Excitation maximum = 485 nm, emission maximum = 535 nm. Longer peptide version, FAM-DEALAHypYIPMDDDFQLRSF, also available.
T41173 FAM-DEALAHypYIPMDDDFQLRSF

Others Others
FAM-DEALAHypYIPMDDDFQLRSF is a 5,6-carboxyfluorescein (FAM) labeled HIF-1α peptide. It binds with high affinity to von Hippel-Lindau (VHL) protein (KD= 3 nM). Can be used to assess ligand binding to VHL in a direct fluorescence polarization (FP) displacement assay. Excitation/emission maxima (λ) = 485/520 nm. This product is a longer peptide version of FAM-DEALA-Hyp-YIPD.

化合物

DEALA-Hyp-YIPD
Cat.No: T82595
Synonym:
Target:
FAM-DEALA-Hyp-YIPD
Cat.No: T41172
Synonym:
Target:
FAM-DEALAHypYIPMDDDFQLRSF
Cat.No: T41173
Synonym:
Target: Others
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