Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5402 |
DDR1-IN-2
DDR1 inhibitor 7rh |
Discoidin Domain Receptor (DDR) | Tyrosine Kinase/Adaptors |
DDR1-IN-2 (DDR1 inhibitor 7rh) 是盘状结构域受体 1 抑制剂 (IC50:13.1 nM),对 DDR2 的抑制作用相对较弱 (IC50:203 nM)。 | |||
T70201 |
S 16020-2
|
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S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors. | |||
T79811 |
DDR1/2 inhibitor-2
|
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DDR1/2 inhibitor-2 (Example 31),作为一种DDR1/DDR2抑制剂,其IC50值小于100 nM,适用于癌症和纤维化疾病的研究领域。 |