Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6453 |
Conivaptan hydrochloride
Vaprisol,盐酸考尼伐坦,Conivaptan HCl,YM 087 |
Vasopressin Receptor | GPCR/G Protein |
Conivaptan hydrochloride (Vaprisol) 是一种口服有效的加压素 V2 和 V1A 受体拮抗剂,用于治疗高血容量性低钠血症和正常血容量。 | |||
T21378 |
Conivaptan
YM087,YM-087,YM 087,Vaprisol |
||
Conivaptan, a non-peptide inhibitor of antidiuretic hormone, was approved for hyponatremia caused by the syndrome of inappropriate antidiuretic hormone (SIADH), there is also some evidence that it may be effective in heart failure. Conivaptan inhibits sub |