首页 工具
登录
购物车

搜索结果

Search Results for " combretastatin a 4 "

6

抑制剂 & 化合物

1

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T31857 Fosbretabulin [free base]

Fosbretabulin,Combretastatin A-4,CA4DP

Fosbretabulin is a natural cis-stilbene that interferes with cellular tubulin dynamics and selectively destroys tumor blood vessels.
T32127 HYS-32

HYS 32

HYS-32, as an analog of combretastatin A-4, can exert by enhancing connexin43 expression.
T60823 isoCA-4

isoCA-4 是一种 Combretastatin A4 的衍生物。 isoCA-4 是一种微管蛋白聚合抑制剂, 具有抗增殖活性。
T35251 YK-5-252

YK 5 252,YK5-252,YK-5252

YK-5-252 is a dual action combretastatin A-4 (CA-4) prodrug which releases CA-4 through a disulfide bond cleavage mechanism and contains a near-infrared (NIR) fluorophore.
T68400 STA-9584

STA-9584 is a potent vascular disrupting agent, which exhibits potent antitumor activity by selectively targeting microvasculature at both the center and periphery of tumors. In vitro, 2-methoxy-5-(5-(3,4,5-trimethoxyphenyl)isoxazol-4-yl)aniline (STA-9122) (active metabolite of STA-9584 ) displayed increased potency relative to other tubulin-binding agents and was highly cytotoxic to tumor cells. STA-9584 induced significant tumor regressions in prostate and breast xenograft models in vivo and, ...
T16386 Ombrabulin hydrochloride

AVE8062 (hydrochloride),AC7700 (hydrochloride)

Microtubule Associated Cytoskeletal Signaling
Ombrabulin hydrochloride 是一种合成的、具有选择性的 CA-4 磷酸酯或 Ombrabulin 的衍生物,能破坏内皮细胞的微管蛋白细胞骨架,具有抗血管作用。Ombrabulin 是是一种微管蛋白聚合抑制剂,是 combretastatin a -4化合物类的一员,是一种水溶性的微管蛋白解聚肿瘤血管破坏化合物。

化合物

Fosbretabulin [free base]
Cat.No: T31857
Synonym: Fosbretabulin,Combretastatin A-4,CA4DP
Target:
HYS-32
Cat.No: T32127
Synonym: HYS 32
Target:
isoCA-4
Cat.No: T60823
Synonym:
Target:
YK-5-252
Cat.No: T35251
Synonym: YK 5 252,YK5-252,YK-5252
Target:
STA-9584
Cat.No: T68400
Synonym:
Target:
Ombrabulin hydrochloride
Cat.No: T16386
Synonym: AVE8062 (hydrochloride),AC7700 (hydrochloride)
Target: Microtubule Associated
Cat. No. Product Name Target Signaling Pathways
T6212 Combretastatin A4

CA4,康普瑞汀,Z)-3,4,5,4',-四甲氧基-3'-羟基二苯乙烯,CRC 87-09

Microtubule Associated Cytoskeletal Signaling
Combretastatin A4 (CA4) 是一种微管靶向剂,可结合 β-tubulin,Kd 值为 0.4 μM。

天然产物

Combretastatin A4
Cat.No: T6212
Synonym: CA4,康普瑞汀,Z)-3,4,5,4',-四甲氧基-3'-羟基二苯乙烯,CRC 87-09
Target: Microtubule Associated
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼