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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14960 |
Chroman 1
|
ROCK | Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells |
Chroman 1 是高效的的ROCK 选择性抑制剂,对 ROCK2 (IC50=1 pM) 的抑制作用强于 ROCK1 (IC50=52 pM) 。它对MRCK 也有抑制作用,IC50为 150 nM。 | |||
T63506 | Chroman 1 dihydrochloride | ||
Chroman 1 dihydrochloride 是选择性的 ROCK 高效抑制剂,对 ROCK2 (IC50: 1 pM) 的作用比 ROCK1 (IC50: 52 pM) 更强,也能够抑制 MRCK 的活性 (IC50: 150 nM)。 | |||
T26086L |
1-((3R,4S)-3-hydroxy-2,2-dimethyl-6-(phenylsulfonyl)chroman-4-yl)pyrrolidin-2-one
|
Others | Others |
1-((3R,4S)-3-hydroxy-2,2-dimethyl-6-(phenylsulfonyl)chroman-4-yl)pyrrolidin-2-one 是 Rilmakalim 的异构体,Rilmakalim 是一种钾通道打开剂 (PCO),可以激活心脏或其它组织中 ATP-敏感 K+ 通道 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1240 |
(2R,3R)-3,7-Dihydroxy-2-(4-hydroxyphenyl)-5-methoxy-8-(3-methylbut-2-en-1-yl)chroman-4-one
3,7,4'-Trihydroxy-5-methoxy-8-prenylflavanone,(2R,3R)-3,7,4'-三羟基-5-甲氧基-8-异戊烯基二氢黄酮 |
Others | Others |
3,7,4'-Trihydroxy-5-methoxy-8-prenylflavanone is a natural product |