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Cat. No. Product Name Target Signaling Pathways
T3338 Ceralasertib

AZD6738

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Ceralasertib (AZD6738) 是一种具有口服活性的选择性 ATR 激酶抑制剂,IC50 为 1 nM。
T26981 Ceralasertib formate

Ceralasertib,AZD-6738,AZD 6738,AZD6738

Ceralasertib is an orally available inhibitor of ataxia telangiectasia and rad3 related (ATR) kinase. Ceralasertib selectively inhibits ATR activity by blocking the downstream phosphorylation of the serine/threonine protein kinase CHK1. This prevents ATR-
T12795 (S)-Ceralasertib

(S)-AZD6738

Others Others
(S)-Ceralasertib is a potent and selective inhibitor of sulfoximine morpholinopyrimidine ATR with excellent preclinical physicochemical and pharmacokinetic (PK) characteristics. .

化合物

Ceralasertib
Cat.No: T3338
Synonym: AZD6738
Target: ATM/ATR
Ceralasertib formate
Cat.No: T26981
Synonym: Ceralasertib,AZD-6738,AZD 6738,AZD6738
Target:
(S)-Ceralasertib
Cat.No: T12795
Synonym: (S)-AZD6738
Target: Others
TargetMol Loading
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