首页 工具
登录
购物车

搜索结果

Search Results for " cyp4a11/cyp4f2-in-1 "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T72501 CYP4A11/CYP4F2-IN-1

P450 Metabolism
CYP4A11/CYP4F2-IN-1 是一种高效的小分子细胞色素 P450 (CYP) 4A11 和 CYP4F2 抑制剂,对P450 (CYP) 4A11 的 IC50 值为 19 nM,对 CYP4F2 的 IC50 值为 17 nM。CYP4A11/CYP4F2-IN-1 可用于研究肾脏疾病和心脑血管疾病。
T36462 CAY10770

CAY10770

CAY10770 is an inhibitor of the cytochrome P450 (CYP) isoform CYP4Z1 (IC50= 5.9 μM).1It is selective for CYP4Z1 over CYP4A11, CYP4F2, CYP4F3a, CYP4F3b (IC50s = 187-282 μM) but does inhibit CYP4F8 and CYP4F12 (IC50s = 167 and 91 μM, respectively). CAY10770 (3 μM) inhibits the production of 14(15)-EET, 19-HETE, and 14(15)-DiHET by 83, 86, and 80%, respectively, in T47D breast cancer cells expressing CYP4Z1. 1.Kowalski, J.P., McDonald, M.G., Pelletier, R.D., et al.Design and characterization of the...

化合物

CYP4A11/CYP4F2-IN-1
Cat.No: T72501
Synonym:
Target: P450
CAY10770
Cat.No: T36462
Synonym: CAY10770
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼