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Cat. No. | Product Name | Target | Signaling Pathways |
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T80421 |
CSD-CH2(1,8)-NH2
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Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
CSD-CH2(1,8)-NH2 是一种针对KOR的选择性且竞争性拮抗剂,具有较低的Ki值(6.8 nM),能够抑制DRG神经元内的钙动员,并能拮抗U50,488的抗伤害效应,常用于神经精神疾病研究领域。 | |||
T11850 |
LIN28 inhibitor LI71
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LIN28 inhibitor LI71 是一种有效的细胞渗透性 LIN28 抑制剂,可消除 LIN28 介导的寡尿苷酸化,IC50 为 7 uM。它能直接绑定 CSD,抑制 LIN28 对 let-7 的作用活性。 | |||
T81932 |
LIN28-IN-1
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LIN28-IN-1(compound 5)是针对RNA结合蛋白LIN28的抑制剂,可与LIN28的冷休克结构域(CSD)发生结合。该化合物能有效阻断LIN28与let-7miRNA的交互作用,具有显著的IC50值为5.4 μM,从而抑制LIN28在表观遗传学中的负向调控功能。此外,LIN28-IN-1在IC50为6.4 μM的条件下,显著抑制了过表达LIN28的JAR癌细胞的增殖。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-01009 |
TGFBI Protein, Human, Recombinant (His)
CDG2,CSD,EBMD,CSD1,CDGG1,CSD3,tra... |
Human | HEK293 Cells |
TGFBI is an RGD-containing protein that binds to type I, II and IV collagens. The RGD motif is found in many extracellular matrix proteins modulating cell adhesion and serves as a ligand recognition sequence for several integrins. TGFBI plays a role in cell-collagen interactions and may be involved in endochondral bone formation in cartilage. TGFBI is induced by transforming growth factor-beta and acts to inhibit cell adhesion. Mutations in TGFBI are associated with multiple types of corneal dys... |