Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79655 |
CRM1-IN-2
|
CRM1 | Membrane transporter/Ion channel |
CRM1-IN-2(Compound KL2)为非共价CRM1抑制剂,能够定位CRM1于核外围,耗尽核内CRM1,从而抑制CRM1介导的核输出。该化合物能抑制结直肠癌细胞的生长并诱导细胞凋亡(apoptosis)。 |