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抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T60050 ANT3310

Antibacterial Microbiology/Virology
ANT3310 是一种广谱共价丝氨酸 β-内酰胺酶抑制剂,对 AmpC、CTX-M-15、TEM-1、OXA-48、OXA-23 和 KPC-2 的 IC50 范围为 1 nM 至 175 nM。 ANT3310 可用于细菌感染研究。
T34671 SNIPER(CRABP)-11

SN 11,SN11,SN-11

SNIPER(CRABP)-11 is a potent protein degrader. SNIPER(CRABP)-11 displayed degradation activity toward the mitochondrial CRABP-II protein.
T13838 PROTAC CRABP-II Degrader-3

Others Others
PROTAC CRABP-II Degrader-3 is a potent degrader of cellular retinoic acid binding protein (CRABP-II) based on cIAp1.
T13836 PROTAC CRABP-II Degrader-1

Others Others
PROTAC CRABP-II Degrader-1 is a potent degrader of cellular retinoic acid binding protein (CRABP-II) based on cIAp1.
T13837 PROTAC CRABP-II Degrader-2

Others Others
PROTAC CRABP-II Degrader-2 is a potent degrader of cellular retinoic acid binding protein (CRABP-II) based on cIAp1.
TP1861L Gly-Phe-Arg acetate(121822-47-7 free base)

Others Others
Gly-Phe-Arg acetate(121822-47-7 free base) 是一种模拟泥蟹抽吸信息素的超强合成三肽。
TP1861 Gly-Phe-Arg

Gly-Phe-Arg is a highly potent synthetic tripeptide that mimics the pumping pheromone of the mud-crab.
T32602 Laurylsarcosyltaurine

Lauryl-sar-taurine

Laurylsarcosyltaurine is a surface active constituent of crab gastric juice.
T35756 Avermectin B1a monosaccharide

Avermectin B1a monosaccharide is a macrolide anthelmintic and monosaccharide form of avermectin B1a . It is lethal to C. elegans with a minimum active concentration (MAC) value of 0.1 μM. Avermectin B1a monosaccharide also stimulates conductance in isolated shore crab muscle.
T83744 Tiger17 TFA

H-Trp-Cys-Lys-Pro-Lys-Pro-Lys-Pro-Arg-Cys-His-NH2

Tiger17是一种环状肽,属于tigerinin-RC1和tigerinin-RC2的衍生物,这两种化合物是在螃蟹吃蛙(F. cancrivora)皮肤分泌物中发现的抗微生物肽。在5至20µg/ml的浓度范围内使用时,Tiger17能增加HaCaT角质形成细胞和人类皮肤成纤维细胞的增殖,并且在20µg/ml的浓度下增加HaCaT细胞的迁移。此外,Tiger17还能增加RAW 264.7巨噬细胞的招募及其TGF-β1和IL-6的分泌。在全层皮肤创伤的小鼠模型中,局部应用20µg/ml的Tiger17能加速伤口闭合和重新上皮化的速度。

化合物

ANT3310
Cat.No: T60050
Synonym:
Target: Antibacterial
SNIPER(CRABP)-11
Cat.No: T34671
Synonym: SN 11,SN11,SN-11
Target:
PROTAC CRABP-II Degrader-3
Cat.No: T13838
Synonym:
Target: Others
PROTAC CRABP-II Degrader-1
Cat.No: T13836
Synonym:
Target: Others
PROTAC CRABP-II Degrader-2
Cat.No: T13837
Synonym:
Target: Others
Gly-Phe-Arg acetate(121822-47-7 free base)
Cat.No: TP1861L
Synonym:
Target: Others
Gly-Phe-Arg
Cat.No: TP1861
Synonym:
Target:
Laurylsarcosyltaurine
Cat.No: T32602
Synonym: Lauryl-sar-taurine
Target:
Avermectin B1a monosaccharide
Cat.No: T35756
Synonym:
Target:
Tiger17 TFA
Cat.No: T83744
Synonym: H-Trp-Cys-Lys-Pro-Lys-Pro-Lys-Pro-Arg-Cys-His-NH2
Target:
Cat. No. Product Name Target Signaling Pathways
T22291 Chitin

Chitin (From shrimp and crab shells)

Others Others
Chitin 是一种大型的结构多糖,存在于真菌的细胞壁、昆虫的外骨骼以及鱼类和无脊椎动物的某些坚硬结构中。

天然产物

Chitin
Cat.No: T22291
Synonym: Chitin (From shrimp and crab shells)
Target: Others
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