Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10792L |
CHK1-IN-4 hydrochloride
CHK1-IN-4 hydrochloride(2120398-41-4 Free base) |
Chk | Cell Cycle/Checkpoint |
CHK1-IN-4 hydrochloride 是有效的checkpoint kinase 1 (chk1) 抑制剂,对肿瘤细胞中 chk1 磷酸化具有有效的抑制作用。CHK1-IN-4 hydrochloride 显示出抗肿瘤活性。 | |||
T10792 |
CHK1-IN-4
|
Chk | Cell Cycle/Checkpoint |
CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity. | |||
T82393 | FLT3/CHK1-IN-1 | ||
FLT3/CHK-IN-1(Compound 18)为FLT3/CHK1双重抑制剂,其对c-KIT的选择性超1700倍,同时显著降低对hERG的亲和力,IC50为58.4 μM。在MV-4-11细胞接种小鼠异种移植模型中有效抑制肿瘤生长。 |