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Cat. No. Product Name Target Signaling Pathways
T14945 CH-0793076

TP3076

Topoisomerase DNA Damage/DNA Repair
CH-0793076, a hexacyclic camptothecin analog, is an active drug and major metabolite of TP300. CH-0793076 is efficacious against cells expressing BCRP (breast cancer resistance protein). CH-0793076 inhibits DNA topoisomerase I (IC50: 2.3 μM).
T73672 CH-0793076 TFA

CH-0793076 (TP3076) TFA,喜树碱的六环类似物,是 TP300 的活性药物和主要代谢物。CH-0793076 TFA 抑制 DNA 拓扑异构酶 I (DNAtopoisomeraseI),IC50为 2.3 μM。CH-0793076 TFA 对表达 BCRP(乳腺癌耐药蛋白) 的细胞也有活性。
T13191 TP3011

CH0793011

Others Others
TP3011 is a potent topoisomerase I inhibitor equipotent as SN38 and is an active metabolite of CH-0793076.

化合物

CH-0793076
Cat.No: T14945
Synonym: TP3076
Target: Topoisomerase
CH-0793076 TFA
Cat.No: T73672
Synonym:
Target:
TP3011
Cat.No: T13191
Synonym: CH0793011
Target: Others
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