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Cat. No. Product Name Target Signaling Pathways
T39247 CDK7-IN-5

CDK7-IN-5

CDK7-IN-5, a CDK7 inhibitor with an IC 50 value of less than 100 nM, exhibits potent anticancer properties (WO2015154022A1, Compound 104).
T39372 CDK7-IN-1

CDK7-IN-1

CDK7-IN-1 is an analog derived from YKL-5-124 and functions as an inhibitor of cyclin-dependent kinase 7 (cdk7). It exhibits strong inhibitory activity, with an IC50 value of less than 100 nM (WO 2016105528 A2, Compound 215).
T16784 Roniciclib

BAY 1000394

CDK Cell Cycle/Checkpoint
Roniciclib (BAY 1000394) 是一种有效的泛 CDK 抑制剂和新型口服细胞毒剂,对 CDK1、CDK2、CDK3、CDK4、CDK7CDK9 的 IC50值为 5-25 nM。

化合物

CDK7-IN-5
Cat.No: T39247
Synonym: CDK7-IN-5
Target:
CDK7-IN-1
Cat.No: T39372
Synonym: CDK7-IN-1
Target:
Roniciclib
Cat.No: T16784
Synonym: BAY 1000394
Target: CDK
TargetMol Loading
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