Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10740 |
CDK8-IN-1
|
CDK | Cell Cycle/Checkpoint |
CDK8-IN-1 是一个有效的、CDK8 的选择性抑制剂,其 IC50 值为 3 nM。 | |||
T10739 | CDK8/19-IN-1 | CDK | Cell Cycle/Checkpoint |
CDK8/19-IN-1 is a selective and oral bioavailable CDK8/19 dual inhibitor (IC50s: 0.46 nM, 0.99 nM, and 270 nM for CDK8, CDK19, and CDK9). |