Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14990 |
CDK12-IN-3
|
CDK | Cell Cycle/Checkpoint |
CDK12-IN-3 is a selective CDK12 inhibitor (IC50: 491 nM in an enzymatic assay). | |||
T62926 |
CDK7/12-IN-1
|
||
CDK7/12-IN-1 是一种 CDK7/12 的选择性抑制剂,作用于 CDK7 (IC50: 3 nM) 和 CDK 12 (IC50: 277 nM)。抑制 CDK7 和 CDK12 是一种有效抑制肿瘤生长的有效。 |