Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12345 |
CBP/p300-IN-3
P300/CBP-IN-3 |
Histone Acetyltransferase | Chromatin/Epigenetic |
CBP/p300-IN-3 (P300/CBP-IN-3) 是一种组蛋白乙酰转移酶抑制剂。 | |||
T63110 |
CBP/p300-IN-15
|
||
CBP/p300-IN-15 (compound 13a) 是一种有效的 p300 (IC50: 2.5 nM) 和 CBP (IC50: 28.0 nM) 抑制剂。CBP/p300-IN-15 能够较好的抑制 OVCAR-3 细胞 (EC50: 0.865 μM) 和 A2780 细胞 (EC50: 2.71 μM)。 CBP/p300-IN-15 能够用于研究卵巢癌。 |