Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79007 |
CARM1-IN-3
|
Histone Methyltransferase | Chromatin/Epigenetic |
CARM1-IN-3 (compound 17b) 是一种针对co-activator associated argininemethyltransferase (CARM1)的高效选择性抑制剂,其IC50值为 0.07 µM。 | |||
T63180 | CARM1-IN-3 dihydrochloride | ||
CARM1-IN-3 dihydrochloride (compound 17b) CARM1-IN-3二盐酸盐(化合物17b)是一种强效的、选择性辅助共激活因子相关的精氨酸甲基转移酶(CARM1)抑制剂,能够作用于 CARM1 (IC50: 0.07 μM)和 CARM3 (IC50>25 μM)。 |