Cat. No. | Product Name | Target | Signaling Pathways |
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T75789 |
CALP3 TFA
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CALP3 TFA 是一种模拟 Ca2+ 的有效肽类 Ca2+ 通道阻断剂,能够激活 EF 手的 Ca2+ 结合蛋白。它通过影响钙调蛋白 (CaM)、Ca2+ 通道及泵的功能来模拟 [Ca2+]i 的增加,从而具备在控制 HIV 或缺血性神经元损伤等情况下调控细胞凋亡的能力。 | |||
TP2170 |
CALP3 TFA(261969-05-5 free base)
CALP3 TFA |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
CALP3 TFA is a potent Ca2+ channel blocker that activates EF-hand motifs of Ca2+-binding proteins. It can functionally mimic increased [Ca2+]i by modulating the activity of Calmodulin, Ca2+ channels, and pumps. |